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Netarsudil (dimesylate) | 奈他地尔甲磺酸
MCE 国际站:Netarsudil (dimesylate)
中文名:奈他地尔甲磺酸
CAS:1422144-42-0
品牌:MedChemExpress (MCE)
存储条件:Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
生物活性:Netarsudil mesylate (AR-13324 mesylate) 甲磺酸盐是ROCK激酶和去甲肾上腺素转运体抑制剂。
热销产品:5(6)-ROX | DBCO-PEG4-Maleimide | Palmitoylethanolamide | Atomoxetine (hydrochloride) | Lenacapavir | Neurofascin, Human (HEK293, His) | ALX-5407 (hydrochloride) | SGC-AAK1-1 | VLX600 | Biotin-PEG2-azide
研究领域:Cell Cycle/DNA Damage | Stem Cell/Wnt | Cytoskeleton | TGF-beta/Smad
作用靶点:ROCK
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides
参考文献:[1]. Wang RF, et al. Effect of 0.04% AR-13324, a ROCK, and norepinephrine transporter inhibitor, on aqueous humor dynamics in normotensive monkey eyes. J Glaucoma. 2015 Jan;24(1):51-4.[2]. Levy B, et al. Ocular hypotensive safety and systemic absorption of AR-13324 ophthalmic solution in normal volunteers. Am J Ophthalmol. 2015 May;159(5):980-5.e1.
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