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Fosaprepitant (dimeglumine) | 福沙吡坦二甲葡胺
MCE 国际站:Fosaprepitant (dimeglumine)
中文名:福沙吡坦二甲葡胺
CAS:265121-04-8
品牌:MedChemExpress (MCE)
存储条件:4°C, sealed storage, away from moisture
生物活性:Fosaprepitant dimeglumine (MK-0517) 是 Aprepitant (HY-10052) 的前药。 Fosaprepitant dimeglumine 是一种神经激肽-1 受体拮抗剂,正在开发用于预防化疗引起的恶心和呕吐 (CINV)[1]。 IC50 和目标:神经激肽-1 受体[1]
体内:Fosaprepitant dimeglumine(30 mg/kg;腹腔注射;每天;持续 7 天)在大鼠中减弱对吗啡的耐受性并增加抗伤害作用[1]。
热销产品:Ajmaline | Atropine (sulfate monohydrate) | Melittin (TFA) | VX-11e | TCIP 1 | Sonelokimab | 1-Methyluric acid | Pyridoxal 5'-phosphate (monohydrate) | Prednisone acetate | Pronethalol
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Neurokinin Receptor
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides
参考文献:[1]. Pranav Prasoon, et al. Role of fosaprepitant, a neurokinin Type 1 receptor antagonist, in morphine-induced antinociception in rats. Indian J Pharmacol. 2016 Jul-Aug; 48(4): 394-398.
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