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STM——内体NK1R信号通路是缓解疼痛的高效靶点
STM—内体NK1R信号通路是缓解疼痛的高效靶点
1.NK1R endocytosis-dependent compartmentalized signaling.
2.G protein–dependent NK1R signaling in endosomes.
3.NK1R endocytosis and neuronal excitation in spinal cord slices.
4.NK1R endocytosis, 1R pERK NeuN ERK signaling, and nociception in vivo.
5.Disruption of NK1R/bARR interactions.
6.Antagonism of endosomal NK1R.
7.Antagonism of endosomal NK1R in spinal cord slices and in vivo.
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