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MCE 国际站:Insulin degludec
CAS:844439-96-9
品牌:MedChemExpress (MCE)
存储条件:Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性:德谷胰岛素是一种超长效形式的胰岛素,用于治疗由 1 型和 2 型糖尿病引起的高血糖症。 Insulin degludec 显示结合效率,对胰岛素受体的 IC50 值为 19.59 nM/L。 Insulin degludec可用于1型和2型糖尿病的研究[1][2]。 IC50 和目标:IC50:19.59 nM/L(胰岛素受体)[2]
体外:Cyclizine抑制离体人肺片段抗ige诱导的组胺释放,IC50为5.42µM[2]。
体内:Insulin degludec(5 U/kg;每天皮下注射一次,持续 30 天)影响胰岛素诱导的低血糖症糖尿病小鼠的葡萄糖稳态和肝脏代谢[1]。
热销产品:PNU-74654 | L-Homocitrulline | L-Threonine | Gymnemic acid I | IA-Alkyne | Cipemastat | Mivacurium (dichloride) | Netupitant | BCTC | ML-193
研究领域:Protein Tyrosine Kinase/RTK
作用靶点:Insulin Receptor
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides
参考文献:[1]. Bataglini C, et al. Insulin degludec and glutamine dipeptide modify glucose homeostasis and liver metabolism in diabetic mice undergoing insulin-induced hypoglycemia. J Appl Biomed. 2021 Dec;19(4):210-219.
[2]. Hartmann T, et al. Effect of the long-acting insulin analogues glargine and degludec on cardiomyocyte cell signalling and function. Cardiovasc Diabetol. 2016 Jul
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