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国际站:Leukotriene B4
CAS:71160-24-2
品牌:MedChemExpress (MCE)
存储条件:Solution, -20°C, 2 years
生物活性:白三烯 B4 (LTB4) 被认为是最有效的化学引诱剂和白细胞激活剂之一,与炎症性疾病有关。白三烯 B4 也是一种基于烷基链的 PROTAC 接头,可用于 PROTAC 的合成[1][2][3] 。
体外:白三烯 B4 诱导中性粒细胞、单核细胞和嗜酸性粒细胞的募集和激活。它还能刺激多种促炎细胞因子和介质的产生,表明其具有增强和延长组织炎症的能力[2]。白三烯 B4 是一种在骨髓细胞中合成的促炎介质,来自花生四烯酸[2].
参考文献:[1]. An S, et al. Small-molecule PROTACs: An emerging and promising approach for the development of targeted therapy drugs. EBioMedicine. 2018 Oct;36:553-562[2]. S.WCrooks, et al. Leukotriene B4. The International Journal of Biochemistry & Cell Biology Volume 30, Issue 2, 27 March 1998, Pages 173-178.[3]. Takehiko Yokomizo, et al. Leukotriene B4: Metabolism and Signal Transduction. Archives of Biochemistry and Biophysics Volume 385, Issue 2, 15 January 2001, Pages 231-241.
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